synthesis and antimicrobial activity of some novel heterocycles containing thiazole, oxazole, thiazine, oxazine and triazole moiety

نویسندگان

vijay v. dabholkar

organic research laboratory, department of chemistry, kc college, churchgate, mumbai, india sunil r. patil

organic research laboratory, department of chemistry, kc college, churchgate, mumbai, india rajesh v. pandey

organic research laboratory, department of chemistry, kc college, churchgate, mumbai, india

چکیده

indandione 1 was brominated to yield 2-bromoindandione 2 which on further reacted with substituted thiocarbamides, carbamides, 2-aminothiophenols, 2-aminophenol and triazoles to furnished 3-substituted aniline-2-thia-4-aza-6,7-benzo-8-oxo-bicyclo [3.3.0]-1(5),3-octadiene 3, 3-substituted aniline-2-oxa-4-aza-6,7-benzo-8-oxo-bicyclo [3.3.0]-1(5),3-octadiene 4, 2-thia-5-aza-9-oxo-3,4-(3’-substituted) benzo-7,8-benzo-bicyclo [4.3.0]-1(6) nonene 5, 2-oxa-5-aza-9-oxo-(3, 4)-(7, 8)-dibenzo-bicyclo [4.3.0]-1(6) nonene 6, 3-substituted-(1,2,4) triazolo [4,5-b] [indeno (2,3-e)]-1,3,4-thiadiazine 7 respectively.

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منابع مشابه

Synthesis and antimicrobial activity of some novel heterocycles containing thiazole, oxazole, thiazine, oxazine and triazole moiety

Indandione 1 was brominated to yield 2-bromoIndandione 2 which on further reacted with substituted thiocarbamides, carbamides, 2-aminothiophenols, 2-aminophenol and triazoles to furnished 3-substituted aniline-2-thia-4-aza-6,7-benzo-8-oxo-bicyclo [3.3.0]-1(5),3-octadiene 3, 3-substituted aniline-2-oxa-4-aza-6,7-benzo-8-oxo-bicyclo [3.3.0]-1(5),3-octadiene 4, 2-Thia-5-aza-9-oxo-3,4-(3’-substitut...

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عنوان ژورنال:
journal of the iranian chemical research

جلد ۴، شماره ۱، صفحات ۳۳-۳۸

کلمات کلیدی
[ ' m o n o b r o m o i n d a n d i o n e ' , ' t h i o c a r b a m i d e ' , ' c a r b a m i d e ' , 2 , ' a m i n o t h i o p h e n o l ' , 2 , ' a m i n o p h e n o l ' , ' t r i a z o l e ' ]

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